Trk Receptor Inhibitors

TrkA

TrkB

TrkC

Trk

Trk Receptor Inhibitors, Agonists, Antagonists, Activators, Modulators, Degraders & Ligands

Product Name	TrkA	TrkB	TrkC	Trk	Purity
ANA-12		TrkB			99.90%
Larotrectinib	TrkA	TrkB	TrkC		99.93%
7,8-Dihydroxyflavone		TrkB			99.74%
Repotrectinib	TrkA				99.95%
TrkA/NGF-IN-1	TrkA				98.22%
TrkA-IN-5	TrkA, IC₅₀: 1.678 nM
N-Acetyl-5-hydroxytryptamine		TrkB			99.96%
GW 441756	TrkA, IC₅₀: 2 nM				99.85%
Amitriptyline	TrkA	TrkB			99.94%
Sitravatinib	TrkA, IC₅₀: 5 nM	TrkB, IC₅₀: 9 nM			99.57%
Amitriptyline hydrochloride	TrkA	TrkB			99.94%
LM22B-10		TrkB	TrkC		99.92%
Cyclotraxin B		TrkB			99.78%
Selitrectinib	TrkA, IC₅₀: 0.6 nM		TrkC, IC₅₀: <2.5 nM		99.90%
Lestaurtinib	TrkA, IC₅₀: 25 nM				99.66%
GNF-5837	TrkA, IC₅₀: 11 nM	TrkB, IC₅₀: 9 nM	TrkC, IC₅₀: 7 nM		99.44%
Altiratinib	Trk1, IC₅₀: 0.85 nM	Trk2, IC₅₀: 4.6 nM	Trk3, IC₅₀: 0.93 nM		99.29%
Larotrectinib sulfate	TrkA	TrkB	TrkC		99.02%
Tamnorzatinib	TrkA				98.59%
Ganglioside GM1	TrkA				99.0%
Tavilermide	TrkA				99.57%
AZ-23	TrkA, IC₅₀: 2 nM	TrkB, IC₅₀: 8 nM			98.92%
Tyrphostin AG 879	TrkA				99.26%
HIOC		TrkB			99.94%
Belizatinib	TrkA	TrkB	TrkC		99.62%
PF-06273340	TrkA, IC₅₀: 6 nM	TrkB, IC₅₀: 4 nM	TrkC, IC₅₀: 3 nM		98.8%
PF-6683324	TrkA, IC₅₀: 1.9 nM (in cell-based assays)	TrkB, IC₅₀: 2.6 nM (in cell-based assays)	TrkC, IC₅₀: 1.1 nM (in cell-based assays)		99.41%
TrkA-IN-3	TrkA, IC₅₀: 22.4 nM				98.01%
Cannflavin B		TrkB			98.36%
Amitriptyline hydrochloride (Standard)	TrkA	TrkB
Zurletrectinib	TrkA, IC₅₀: 0.81 nM	TrkB, IC₅₀: 0.145 nM	TrkC, IC₅₀: 0.184 nM		99.32%
Paltimatrectinib	TrkA				99.95%
CG428	TrkA, Kd: 1 nM	TrkB, Kd: 28 nM	TrkC, Kd: 4.2 nM		98.26%
TrkA-IN-4	TrkA				98.99%
Levomilnacipran hydrochloride		TrkB			99.95%
PF-06737007	TrkA, IC₅₀: 7.7 nM (in cell-based assays)	TrkB, IC₅₀: 15 nM (in cell-based assays)	TrkC, IC₅₀: 3.9 nM (in cell-based assays)		99.90%
DS-1205b free base	TrkA, IC₅₀: 407 nM				99.92%
TrkA-IN-1	TrkA, IC₅₀: 99 nM	TrkB, IC₅₀: 81 μM	TrkC, IC₅₀: 25 μM
CH7057288				TRK	99.73%
CE-245677	TrkA				98.00%
ZEB85		TrkB
MNAC13	TrkA
FLY26		TrkB			99.66%
CZS-241	TrkA, IC₅₀: 2.74 μM
Sitravatinib malate	TrkA, IC₅₀: 5 nM	TrkB, IC₅₀: 9 nM
LPM4870108	TrkA, IC₅₀: 2.4 nM		TrkC, IC₅₀: 0.2 nM
FLT3/TrKA-IN-1	TrkA, IC₅₀: 23.6 nM
PF-06733804	TrkA, IC₅₀: 8.4 nM (in cell-based assays)	TrkB, IC₅₀: 6.2 nM (in cell-based assays)	TrkC, IC₅₀: 2.2 nM (in cell-based assays)
DS002	TrkA
KRC-108	TrkA, IC₅₀: 39 nM
DZX19	TrkA, IC₅₀: 1.32 nM TRKA^G595R, IC₅₀: 16.56 nM TRKA^F589L, IC₅₀: 74.37 nM TRKA^G667C, IC₅₀: 60.18 nM	TrkB, IC₅₀: 2.28 nM	TrkC, IC₅₀: 4.05 nM
TRK-IN-31 hydrochloride				TRK, : 1.8 nM
Trk-IN-7	TrkA, IC₅₀: <25 nM	TrkB, IC₅₀: <5 nM	TrkC, IC₅₀: <25 nM
TRK/ALK-IN-1	TrkA
TrkB activator-1		TrkB
TRK-IN-31				TRK, : 1.8 nM
PTX-BD10-2		TrkB	TrkC
Trk-IN-8	TrkA		TrkC
Trk-IN-20	TrkA, IC₅₀: 1.6 nM	TrkB, IC₅₀: 2.9 nM	TrkC, IC₅₀: 2.0 nM
TRK-IN-23	TrkA, IC₅₀: 0.5 nM TRKA^G595R, IC₅₀: 14 nM TRKA^F589L, IC₅₀: 4.4 nM TRKA^G667C, IC₅₀: 4.8 nM		TrkC, IC₅₀: 9 nM
ZW-18-116	TrkA
GZ-389988	TrkA, IC₅₀: 0.3 nM	TrkB, IC₅₀: 0.1 nM	TrkC, IC₅₀: 0.5 nM
JYP0322	TrkA	TrkB	TrkC
TIY-7	TrkA, IC₅₀: 2.9 nM
Cyclotraxin B TFA		TrkB
Protein kinase inhibitor 5 sulfate hydrate	TrkA, IC₅₀: 1.8 nM
ZW-6-052	TrkA
Multi-kinase-IN-7	TrkA, IC₅₀: 3.59 μM
Pegcantratinib	TrkA
PF-07245303	TrkA, Kd: 2.94 nM	TrkB, Kd: 8.76 nM	TrkC, Kd: 10 nM
Protein kinase inhibitor 5	TrkA, IC₅₀: 1.8 nM
Trk-IN-11	TrkA
(R)-Larotrectinib	TrkA, IC₅₀: 28.5 nM
TrkB-IN-1		TrkB			99.2%
Trk-IN-10	TrkA
TRK II-IN-1	TrkA, IC₅₀: 3.3 nM	TrkB, IC₅₀: 6.4 nM	TrkC, IC₅₀: 4.3 nM
JND4135	TrkA	TrkB	TrkC
Multi-kinase-IN-6	TrkA, IC₅₀: 0.33 μM
Pan-Trk-IN-3	TrkA, IC₅₀: 2 nM	TrkB, IC₅₀: 3 nM	TrkC, IC₅₀: 2 nM
TRK-IN-34	TRKA^G595R, IC₅₀: 0.75 nM TRKA^G667C, IC₅₀: 0.96 nM TRKA^F589L, IC₅₀: 0.44 nM TrkA, IC₅₀: 2.8 nM		TrkC^G623R, IC₅₀: 0.73 nM TrkC^G696A, IC₅₀: 1.3 nM
NPA101.3	TrkA, IC₅₀: 32 nM
TrkC-IN-1			TrkC
NTRK1-ligand-1	NTRK1
Type II TRK inhibitor 1	TrkA		TrkC
D5261	TrkA
IHMT-TRK-284	TrkA, IC₅₀: 10.5 nM	TrkB, IC₅₀: 0.7 nM	TrkC, IC₅₀: 2.6 nM
TRK-IN-33	TrkA
Anizatrectinib	TrkA
NMS-P626	TrkA, IC₅₀: 8 nM	TrkB, IC₅₀: 3 nM	TrkC, IC₅₀: 7 nM
ONO-7579	TrkA
HS-345	TrkA
BNN-20		TrkB

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